SCHEMBL9565015

SCHEMBL9565015

CC(CC(C(=O)N(C)C)(c1ccccc1)c1ccccc1)N1CCC(Nc2nc3cncnc3n2Cc2ccccn2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.35
CHRM1 P11229 2/20 0.35
CHRM3 P20309 2/20 0.35
GPR6 P46095 1/20 0.34
OPRM1 P35372 4/20 0.33
GBA1 P04062 1/20 0.32
CCR5 P51681 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
SLC5A7 Q9GZV3 1/20 0.32
MEN1 O00255 1/20 0.32
PABPC1 P11940 1/20 0.32
KMT2A Q03164 1/20 0.32
DRD4 P21917 1/20 0.32
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564931 0.88 ALDH1A1 (0.34) OPRM1MEN1KMT2ALMNA
SCHEMBL9866590 0.87 OPRM1 (0.43) CHRM2CHRM1CHRM3GPR6OPRM1
SCHEMBL9565024 0.87 LMNA (0.32) LMNACYP1A2CYP2C9CYP2C19WHR1
SCHEMBL9564925 0.84 CHRM2 (0.38) CHRM2CHRM1CHRM3GPR6OPRM1
SCHEMBL9602879 0.76 NOS2 (0.56) MEN1KMT2A
SCHEMBL8207942 0.74 KCNH2 (0.47) CHRM2CHRM1CHRM3OPRM1SIGMAR1
SCHEMBL9564775 0.73 OPRM1 (0.48) CHRM2CHRM1OPRM1SIGMAR1CYP3A4
SCHEMBL9564838 0.73 SSTR5 (0.43) CHRM2CHRM1CHRM3OPRM1SIGMAR1
SCHEMBL9564782 0.73 KCNH2 (0.45) CYP3A4CYP2D6MEN1KMT2ALMNA
SCHEMBL9565053 0.69 KCNH2 (0.57) CHRM2CHRM1CHRM3OPRM1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed