SCHEMBL9565024

SCHEMBL9565024

Cc1ccc(Cn2c(NC3CCN(C(C)CC(C(=O)N(C)C)(c4ccccc4)c4ccccc4)CC3)nc3cncnc32)o1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
WHR1 P49842 1/20 0.30
UBE2M P61081 1/20 0.30
DCUN1D1 Q96GG9 1/20 0.30
CYP46A1 Q9Y6A2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564931 0.90 ALDH1A1 (0.34) LMNA
SCHEMBL9565015 0.87 CHRM2 (0.35) LMNACYP1A2CYP2C9CYP2C19WHR1
SCHEMBL9564774 0.76 ALDH1A1 (0.44) LMNA
SCHEMBL9866590 0.74 OPRM1 (0.43) LMNACYP1A2
SCHEMBL9564990 0.73 NR4A2 (0.40) LMNACYP1A2CYP2C9CYP2C19
SCHEMBL8207942 0.73 KCNH2 (0.47) LMNACYP1A2CYP2C19
SCHEMBL9564775 0.72 OPRM1 (0.48) LMNACYP1A2CYP2C9CYP2C19
SCHEMBL9564808 0.72 HTR2A (0.38) LMNACYP1A2CYP2C19
SCHEMBL9564925 0.72 CHRM2 (0.38) LMNACYP2C19
SCHEMBL9565023 0.70 USP2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed