SCHEMBL9587168

SCHEMBL9587168

CCC1(CC)C=C(n2ccccc2=O)c2cc(Br)ccc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
PTPRC P08575 1/20 0.35
S100A4 P26447 1/20 0.32
APAF1 O14727 1/20 0.32
SMAD3 P84022 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
F10 P00742 1/20 0.31
ALDH1A1 P00352 1/20 0.30
ALDH2 P05091 1/20 0.30
ALDH3A1 P30838 1/20 0.30
CUL4A Q13619 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9589242 0.85 CA1 (0.39) CA1CA2CA4CA7CA9
SCHEMBL9589614 0.83 ABCC9 (0.38) F10
SCHEMBL9588407 0.80 CA1 (0.39) CA1CA2CA4CA7CA9
SCHEMBL9733913 0.72 TDP1 (0.37) PTPRCTDP1L3MBTL1F10MEN1
SCHEMBL9589861 0.72 ALDH1A1 (0.42) L3MBTL1ALDH1A1HRH4
SCHEMBL8085076 0.72 NPSR1 (0.34) PTPRCF10MEN1KMT2AHRH4
SCHEMBL9587001 0.69 CA1 (0.39) CA1CA2CA7CA9HRH4
SCHEMBL9587407 0.69 S100A4 (0.36) S100A4F10
SCHEMBL9736934 0.69 NPSR1 (0.33)
SCHEMBL9590341 0.68 GFER (0.36) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed