SCHEMBL9588407

SCHEMBL9588407

CC1(C)C=C(n2ccccc2=O)c2ccc(Br)cc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
PTPRC P08575 1/20 0.36
S100A4 P26447 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
F10 P00742 1/20 0.32
HRH4 Q9H3N8 1/20 0.31
POLB P06746 2/20 0.31
CYP1A2 P05177 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9589242 0.95 CA1 (0.39) CA1CA2CA4CA7CA9
SCHEMBL9587505 0.81 SLC6A9 (0.33) F10HRH4POLB
SCHEMBL9587196 0.81 ABCC9 (0.47) CA1CA2F10
SCHEMBL9587168 0.80 CA1 (0.37) CA1CA2CA4CA7CA9
SCHEMBL9587001 0.79 CA1 (0.39) CA1CA2CA7CA9HRH4
SCHEMBL9587407 0.79 S100A4 (0.36) S100A4MAPTF10
SCHEMBL9590341 0.77 GFER (0.36) HRH4
SCHEMBL9589861 0.77 ALDH1A1 (0.42) MAPTRAB9AL3MBTL1HRH4CYP1A2
SCHEMBL8085076 0.77 NPSR1 (0.34) PTPRCMEN1MAPTHTTRAB9A
SCHEMBL9590296 0.77 CA1 (0.43) CA1CA2CA4CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed