SCHEMBL9596295

SCHEMBL9596295

O=C(O)c1ccc(CBr)cc1N1C(=O)CCC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 1/20 0.38
MYC P01106 1/20 0.37
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 5/20 0.35
MAPT P10636 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HPGD P15428 3/20 0.35
TP53 P04637 1/20 0.35
ALDH1A1 P00352 3/20 0.35
PKM P14618 1/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
PARP1 P09874 1/20 0.33
KLKB1 P03952 1/20 0.33
CTSB P07858 1/20 0.33
MMP9 P14780 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484252 0.80 PTGS1 (0.50) CA12CA1CA9MAPK1GAA
SCHEMBL6887707 0.78 CA12 (0.48) CA12CA1CA9MAPK1GAA
SCHEMBL317626 0.76 CA12 (0.42) CA12CA1CA9MAPK1GAA
SCHEMBL31653832 0.76 KEAP1 (0.43) CA12CA1CA9MAPK1GAA
SCHEMBL317703 0.76 KEAP1 (0.43) CA12CA1CA9MAPK1GAA
SCHEMBL7769435 0.76 ALDH1A1 (0.41) CA12CA1CA9KDM4EKMT2A
SCHEMBL29981284 0.75 CRHBP (0.43) MAPK1KDM4EKMT2AMAPTHPGD
SCHEMBL1464604 0.75 CA12 (0.41) CA12CA1CA9MAPK1GAA
SCHEMBL610788 0.75 CA12 (0.41) CA12CA1CA9MAPK1GAA
SCHEMBL10627311 0.74 MCL1 (0.42) CA12CA1CA9MAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5248770-A Labels such as fluorescent or radioactive compounds THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-09-28 US disclosed
US-5098996-A Fluorination of compounds for use in diagnosis of nuclear medicine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1992-03-24 US disclosed