SCHEMBL9596387

SCHEMBL9596387

CCC(=O)Nc1ccc2c(c1)C(n1ccccc1=O)C(O)C(C)(C)C2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
POLB P06746 3/20 0.46
MAPT P10636 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 4/20 0.43
KDM4E B2RXH2 3/20 0.43
PDK2 Q15119 1/20 0.43
CASP3 P42574 1/20 0.41
HSD17B10 Q99714 2/20 0.40
NR3C1 P04150 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704051 0.80 RAB9A (0.44) RAB9AALDH1A1NPC1MEN1KMT2A
SCHEMBL9704045 0.80 RAB9A (0.44) RAB9AALDH1A1NPC1MEN1KMT2A
SCHEMBL9588271 0.79 DRD2 (0.34) ALDH1A1MEN1KMT2AMAPTPDK2
SCHEMBL9589012 0.79 ALDH1A1 (0.36) ALDH1A1MEN1KMT2APOLBCYP1A2
SCHEMBL9588012 0.79 IDO1 (0.34) MAPTPDK2
SCHEMBL9587643 0.78 ALDH1A1 (0.32) RAB9AALDH1A1MEN1KMT2APOLB
SCHEMBL9702059 0.78 ALDH1A1 (0.32) RAB9AALDH1A1MEN1KMT2APOLB
SCHEMBL9587842 0.77 MEN1 (0.41) RAB9AALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL9701823 0.77 MEN1 (0.41) RAB9AALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL9588559 0.76 HSD17B1 (0.34) MEN1KMT2AMAPTCYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US claimed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP claimed
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed