SCHEMBL9602565

SCHEMBL9602565

CC(C)(Br)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
AHR P35869 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR2 P34972 6/20 0.34
CNR1 P21554 5/20 0.34
GAA P10253 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TPMT P51580 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803437 0.79 TSHR (0.50) TSHRTP53CYP3A4MEN1KMT2A
SCHEMBL673309 0.79 TSHR (0.50) TSHRTP53CYP3A4AHRMEN1
SCHEMBL45127 0.77 GABRA1 (0.40) TSHRCYP3A4ALDH1A1
SCHEMBL9403849 0.77 TSHR (0.47) TSHRTP53CYP3A4AHRMEN1
SCHEMBL16396157 0.75 ALDH1A1 (0.44) TSHRCYP3A4MEN1KMT2AALDH1A1
SCHEMBL25134468 0.74 TSHR (0.44) TSHRTP53CYP3A4AHRMEN1
SCHEMBL2646961 0.74 TSHR (0.44) TSHRTP53CYP3A4MEN1KMT2A
SCHEMBL4495782 0.74 TSHR (0.44) TSHRTP53CYP3A4AHRMEN1
SCHEMBL15449818 0.74 TSHR (0.44) TSHRTP53CYP3A4AHRMEN1
SCHEMBL11457726 0.74 MEN1 (0.39) TSHRTP53CYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360829-B1 DEHYDROBROMINATION OF SUBSTITUTED ALPHA-HALOCUMENE DOWELANCO (US) 1993-05-26 EP claimed
US-4594467-A DEHYDROBROMINATING ALPH-BROMO-3,5-DICHLORO CUMENE WITH ALKALI METAL HYDROXIDE IN PRESENCE OF PHASE TRANSFER CATALYST BAYER AKTIENGESELLSCHAFT (DE) 1986-06-10 US claimed
EP-0360829-B1 DEHYDROBROMINATION OF SUBSTITUTED ALPHA-HALOCUMENE DOWELANCO (US) 1993-05-26 EP disclosed
EP-0360829-A1 DEHYDROBROMINATION OF SUBSTITUTED ALPHA-HALOCUMENE. DOW CHEMICAL CO (US) 1990-04-04 EP disclosed
US-4861927-A Dehydrohalogenation of ring-halogenated α-halocumenes THE DOW CHEMICAL COMPANY (US) 1989-08-29 US disclosed
WO-1988009319-A1 DEHYDROBROMINATION OF SUBSTITUTED alpha-HALOCUMENE THE DOW CHEMICAL COMPANY (US) 1988-12-01 WO disclosed
US-4760209-A Isopropylation, isomerization, bromination and dehydrobromination BAYER AKTIENGESELLSCHAFT (DE) 1988-07-26 US disclosed
US-4594467-A DEHYDROBROMINATING ALPH-BROMO-3,5-DICHLORO CUMENE WITH ALKALI METAL HYDROXIDE IN PRESENCE OF PHASE TRANSFER CATALYST BAYER AKTIENGESELLSCHAFT (DE) 1986-06-10 US disclosed
US-4594467-A DEHYDROBROMINATING ALPH-BROMO-3,5-DICHLORO CUMENE WITH ALKALI METAL HYDROXIDE IN PRESENCE OF PHASE TRANSFER CATALYST BAYER AKTIENGESELLSCHAFT (DE) 1986-06-10 US disclosed
US-4087473-A Preferential aliphatic halogenation of ar-substituted alkylbenzenes THE DOW CHEMICAL COMPANY (US) 1978-05-02 US disclosed
US-4087473-A Preferential aliphatic halogenation of ar-substituted alkylbenzenes THE DOW CHEMICAL COMPANY (US) 1978-05-02 US disclosed