SCHEMBL9630571

SCHEMBL9630571

CCCCCc1nc(O)c(-c2ccccc2)s1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.53
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TLR8 Q9NR97 1/20 0.45
TLR7 Q9NYK1 1/20 0.45
GCGR P47871 1/20 0.45
GPR84 Q9NQS5 1/20 0.43
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754030 0.77 ALOX5 (0.44) ALOX5
SCHEMBL9754002 0.73 ALOX5 (0.47) ALOX5
SCHEMBL3681457 0.72 TP53 (0.43) ALOX5TP53MAPTSMN1; SMN2GCGR
SCHEMBL7693026 0.71 NPC1 (0.49) ALOX5TP53MAPTSMN1; SMN2TLR8
SCHEMBL27744669 0.71 DHFR (0.47) ALOX5TP53MAPTSMN1; SMN2GCGR
SCHEMBL27629514 0.71 ALOX5 (0.50) ALOX5TP53MAPTSMN1; SMN2GCGR
SCHEMBL8830209 0.70 NPC1 (0.44) ALOX5TP53MAPTSMN1; SMN2
SCHEMBL9629574 0.70 ALOX5 (1.00) ALOX5TP53MAPT
SCHEMBL27913336 0.69 LOXL2 (0.64) TP53MAPTSMN1; SMN2
SCHEMBL8716614 0.69 ALDH1A1 (0.51) TP53MAPTSMN1; SMN2GPR84DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124342-A Antiinflammatory, antiarthritic agents; antiallergens; skin disorders ABBOTT LABORATORIES (US) 1992-06-23 US disclosed
EP-0457803-A4 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS 1991-12-04 EP disclosed
EP-0457803-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1991-11-27 EP disclosed
WO-1990009801-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1990-09-07 WO disclosed
WO-1990009381-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1990-08-23 WO disclosed