SCHEMBL9665493

SCHEMBL9665493

CC(=O)c1cc(F)ccc1N

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.68
FADS1 O60427 1/20 0.50
CES2 O00748 2/20 0.47
CES1 P23141 2/20 0.47
ALDH1A1 P00352 1/20 0.46
HDAC1 Q13547 5/20 0.43
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 2/20 0.41
GFER P55789 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
BRAF P15056 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29467969 1.00 KEAP1 (0.68) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL18070541 0.85 KDM4E (0.53) KEAP1HDAC1KMT2AKDM4EGFER
SCHEMBL30590455 0.83 KEAP1 (0.52) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL1720983 0.83 KEAP1 (0.52) KEAP1FADS1CES2CES1ALDH1A1
Hydrochloric Acid SCHEMBL4049299 0.82 KEAP1 (0.50) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL183930 0.81 KEAP1 (0.70) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL135091 0.81 KEAP1 (1.00) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL29364785 0.81 KEAP1 (1.00) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL31230207 0.81 KEAP1 (0.70) KEAP1FADS1CES2CES1ALDH1A1
SCHEMBL12789530 0.81 BRAF (0.61) KEAP1HDAC1BRAFHDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117550981-B Preparation method of 2-amino-5-fluoro acetophenone 成都工业学院 2024-03-15 CN claimed
CN-117550981-A Preparation method of 2-amino-5-fluoro acetophenone 成都工业学院 2024-02-13 CN claimed
CN-109384683-B Preparation method of 2-amino-5-fluoroacetophenone 杭州科耀医药科技有限公司 2021-09-03 CN claimed
CN-110922315-A Preparation method of Laolatinib intermediate compound 常州工学院 2020-03-27 CN claimed
EP-0195396-B1 5-FLUOROBENZONITRILE DERIVATIVES AND PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF FOR INCREASING THE LEAN MEAT TO FAT RATIO, AND/OR ENHANCING THE GROWTH RATE OF WARM-BLOODED ANIMALS AMERICAN CYANAMID COMPANY (US) 1989-03-01 EP claimed
EP-0195396-A1 5-Fluorobenzonitrile derivatives and pharmacologically acceptable acid addition salts thereof for increasing the lean meat to fat ratio, and/or enhancing the growth rate of warm-blooded animals AMERICAN CYANAMID COMPANY (US) 1986-09-24 EP claimed
US-20260008774-A1 QUINOLINONE AMIDE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS INC (US) 2026-01-08 US disclosed
US-20250368647-A1 NITROGEN CONTAINING CONDENSED 2,3-DIHYDROQUINAZOLINONE COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2025-12-04 US disclosed
WO-2025235686-A1 FLUOROCAMPTOTHECIN COMPOUNDS, CONJUGATES, AND METHODS THEREOF Aarvik Therapeutics, Inc. (US) 2025-11-13 WO disclosed
US-12448369-B2 Quinolinone amide compounds and uses thereof EDGEWISE THERAPEUTICS, INC. (US) 2025-10-21 US disclosed
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2025-06-05 US disclosed
CN-120058540-A Method for preparing halogenated 2-aminobenzophenone by continuous photochemical rearrangement 姚昕辰 2025-05-30 CN disclosed
WO-2025077773-A1 NOVEL TYPE I TOPOISOMERASE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊维康医药有限责任公司 2025-04-17 WO disclosed
US-4656267-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1987-04-07 US disclosed
US-4622065-A HERBICIDES PPG INDUSTRIES, INC. (US) 1986-11-11 US disclosed
US-4614746-A 5-fluorobenzonitrile derivatives for increasing the lean meat to fat ratio and/or enhancing the growth rate of warm-blooded animals AMERICAN CYANAMID COMPANY (US) 1986-09-30 US disclosed
EP-0195396-A1 5-Fluorobenzonitrile derivatives and pharmacologically acceptable acid addition salts thereof for increasing the lean meat to fat ratio, and/or enhancing the growth rate of warm-blooded animals AMERICAN CYANAMID COMPANY (US) 1986-09-24 EP disclosed
US-4555571-A Substituted 2(1H)-quinazolinone-1-alkanoic acids and esters ORTHO PHARMACEUTICAL CORPORATION (US) 1985-11-26 US disclosed
EP-0138491-A2 Substituted 2(1H)-quinazolinone-1-alkanoic acids and esters ORTHO PHARMACEUTICAL CORPORATION (US) 1985-04-24 EP disclosed
US-3987047-A ANORETICS BOEHRINGER INGELHEIM GMBH (DT) 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12448369-B2 Quinolinone amide compounds and uses thereof TNNI3, TNNT2, COQ8A KEAP1 555/4885FADS1 408/4885CES2 894/4885
US-20250368647-A1 NITROGEN CONTAINING CONDENSED 2,3-DIHYDROQUINAZOLINONE COMPOUNDS AS NAV1.8 INHIBITORS SCN8A, SCN2A, SCN5A KEAP1 1018/4885FADS1 2629/4885CES2 3401/4885
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS AKR1C2, AKR1B1, AKR1C1 KEAP1 247/4885FADS1 319/4885CES2 965/4885
US-20260008774-A1 QUINOLINONE AMIDE COMPOUNDS AND USES THEREOF TNNT2, TNNI3, TNNC1 KEAP1 1335/4885FADS1 1586/4885CES2 632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.