SCHEMBL9682641

SCHEMBL9682641

CN1c2ccccc2C(c2ccccc2F)NCC1CNCc1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
CXCR4 P61073 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KMT2A Q03164 7/20 0.33
MEN1 O00255 6/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CYP2C19 P33261 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683424 0.85 CCKBR (0.38) CCKBRL3MBTL1KMT2AMEN1CYP1A2
SCHEMBL9499330 0.81 CCKBR (0.58) CCKBRHDAC1HDAC8HDAC6KMT2A
SCHEMBL9499432 0.74 OPRM1 (0.49) CCKBR
SCHEMBL9500460 0.69 OPRD1 (0.60) CCKBR
SCHEMBL9501463 0.69 LMNA (0.52) CCKBRKMT2AALDH1A1GAAHTT
SCHEMBL9501442 0.68 CCKBR (0.62) CCKBRKMT2AMEN1KDM4EALDH1A1
SCHEMBL9501031 0.67 CCKBR (0.64) CCKBRHTR2ASMN1; SMN2
SCHEMBL3650807 0.62 KMT2A (0.51) CXCR4KMT2AMEN1KDM4EALDH1A1
SCHEMBL11683129 0.60 HTR2C (0.46) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL3652732 0.59 KMT2A (0.51) CXCR4KMT2AMEN1HTR2CHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486271-A2 Cholecystokinin antagonists for treating neurological disorders MERCK & CO. INC. (US) 1992-05-20 EP claimed