SCHEMBL9686606

SCHEMBL9686606

CCOc1nccc2nc(N3CCNCC3)ncc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.43
CYP1A2 P05177 13/20 0.43
HSD17B10 Q99714 12/20 0.43
HPGD P15428 10/20 0.43
CYP3A4 P08684 10/20 0.43
CYP2C9 P11712 9/20 0.43
USP2 O75604 7/20 0.43
CYP2C19 P33261 5/20 0.43
HIF1A Q16665 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TAAR1 Q96RJ0 1/20 0.42
ADRB1 P08588 1/20 0.42
ACHE P22303 1/20 0.42
CASP1 P29466 10/20 0.41
CASP7 P55210 9/20 0.41
GLA P06280 1/20 0.40
CYP2D6 P10635 3/20 0.40
TP53 P04637 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685414 0.80 DRD2 (0.49) ALDH1A1HPGDACHECASP1MAPK1
SCHEMBL31148464 0.76 MAPT (0.42) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL5258581 0.74 ADRB1 (0.52) ALDH1A1HPGDSMN1; SMN2TAAR1ADRB1
SCHEMBL2920903 0.73 CHRNB2 (0.46) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL9685229 0.72 USP19 (0.51) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL9686750 0.72 USP19 (0.44) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL13116676 0.69 HRH4 (0.44)
SCHEMBL9685430 0.68 USP19 (0.48) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL10721643 0.67 ALDH1A1 (0.54) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4
SCHEMBL30423191 0.67 ADRB1 (0.50) ALDH1A1CYP1A2HSD17B10HPGDADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed