SCHEMBL9686750

SCHEMBL9686750

CCn1ccc2nc(N3CCNCC3)ncc2c1=S

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP19 O94966 1/20 0.44
ALDH1A1 P00352 13/20 0.42
HPGD P15428 10/20 0.42
TAAR1 Q96RJ0 1/20 0.41
CYP1A2 P05177 12/20 0.40
HSD17B10 Q99714 12/20 0.40
CYP3A4 P08684 10/20 0.40
CYP2C9 P11712 8/20 0.40
CYP2C19 P33261 7/20 0.40
USP2 O75604 6/20 0.40
HIF1A Q16665 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CASP1 P29466 10/20 0.39
CASP7 P55210 8/20 0.39
GLA P06280 1/20 0.39
CYP2D6 P10635 3/20 0.39
TSHR P16473 3/20 0.39
MAPK1 P28482 2/20 0.39
ADRB1 P08588 1/20 0.39
HRH4 Q9H3N8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685229 0.88 USP19 (0.51) USP19ALDH1A1HPGDCYP1A2HSD17B10
SCHEMBL9685430 0.76 USP19 (0.48) USP19ALDH1A1HPGDCYP1A2HSD17B10
SCHEMBL10678247 0.76 CASP1 (0.47) ALDH1A1HPGDCYP1A2HSD17B10CYP3A4
Hydrochloric Acid SCHEMBL10508297 0.75 CASP1 (0.47) ALDH1A1HPGDCYP1A2HSD17B10CYP3A4
SCHEMBL9686606 0.72 ALDH1A1 (0.43) ALDH1A1HPGDTAAR1CYP1A2HSD17B10
SCHEMBL9686858 0.71 HTR3A (0.55) USP19ALDH1A1HPGDCYP1A2HSD17B10
SCHEMBL9684556 0.69 LMNA (0.51) ALDH1A1HPGDHSD17B10SMN1; SMN2CASP1
SCHEMBL9686198 0.68 TSHR (0.40) USP19TSHRKMT2AMEN1
SCHEMBL10048250 0.68 CASP1 (0.57) ALDH1A1HPGDCYP1A2HSD17B10CYP3A4
SCHEMBL9685325 0.68 CYP1A2 (0.46) USP19ALDH1A1HPGDCYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed