SCHEMBL9686858

SCHEMBL9686858

CCn1ccc2nc(N3CCN(c4ncc5ccccc5n4)CC3)ncc2c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.55
HRH4 Q9H3N8 1/20 0.55
HCAR2 Q8TDS4 1/20 0.44
HCRTR1 O43613 5/20 0.43
HCRTR2 O43614 5/20 0.43
OGA O60502 1/20 0.43
HTR1A P08908 3/20 0.43
DRD2 P14416 3/20 0.43
HTR2A P28223 3/20 0.43
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
USP19 O94966 1/20 0.41
CASP1 P29466 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.40
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9684556 0.85 LMNA (0.51) HTR1ADRD2HTR2AALDH1A1HSD17B10
SCHEMBL9685229 0.83 USP19 (0.51) ALDH1A1HSD17B10MEN1HPGDKMT2A
SCHEMBL9686198 0.81 TSHR (0.40) MEN1KMT2AUSP19TSHR
SCHEMBL9686141 0.75
SCHEMBL10824274 0.74 NPC1 (0.48) ALDH1A1KDM4EHPGDCASP1LMNA
SCHEMBL9685451 0.73 ADRA2A (0.57)
SCHEMBL27896727 0.72 HTR3A (0.71) HTR3AHRH4HCAR2HCRTR1HCRTR2
SCHEMBL603314 0.72 HTR3A (1.00) HTR3AHRH4HCAR2HCRTR1HCRTR2
SCHEMBL10885460 0.72 BRD9 (0.68) ALDH1A1HSD17B10MEN1HPGDKMT2A
Hydrochloric Acid SCHEMBL9686615 0.71 ADRA1A (0.49) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed