SCHEMBL9687223

SCHEMBL9687223

O=c1ccc(-c2ccc3[nH]c(CCNC(O)C(O)Cc4cccc5ccccc45)nc3c2)n[nH]1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.34
PIK3CB P42338 2/20 0.34
HTT P42858 2/20 0.33
GPR119 Q8TDV5 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
PDE10A Q9Y233 1/20 0.33
MME P08473 2/20 0.33
ECE1 P42892 2/20 0.33
THRB P10828 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7303875 0.83 MAPT (0.41) MEN1KMT2AMMEECE1
SCHEMBL7299013 0.81 DYRK1A (0.37) HTTGPR119MEN1KMT2AEGFR
SCHEMBL7295525 0.78 PDE3B (0.40) GPR119
SCHEMBL9687230 0.77 MAPK1 (0.45) HTTCYP2C9
SCHEMBL7304445 0.74 PDE3B (0.39) GPR119
SCHEMBL7303724 0.71 RAD52 (0.43) GPR119MEN1KMT2ACYP2C9PDE10A
SCHEMBL9688183 0.68 CTSS (0.48) MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL7331760 0.64 SMN1; SMN2 (0.40) GPR119KMT2AMMEECE1
SCHEMBL7303740 0.63 RAD52 (0.52) GPR119MEN1KMT2AKDM4E
SCHEMBL8043227 0.61 EGFR (0.55) HTTMEN1KMT2AEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed