SCHEMBL9688670

SCHEMBL9688670

COc1ccc(CCN(C)C)c(N)c1N

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 4/20 0.50
HTR2A P28223 1/20 0.47
HTR1A P08908 1/20 0.46
NOS1 P29475 2/20 0.45
HTR6 P50406 2/20 0.44
NOS3 P29474 1/20 0.42
ACHE P22303 1/20 0.40
MDM2 Q00987 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688926 0.81 HTR1A (0.46) AOC3HTR1A
SCHEMBL2939712 0.78 GAA (0.40) AOC3
SCHEMBL4360488 0.77 AOC3 (0.55) AOC3HTR2AHTR1ANOS1NOS3
SCHEMBL9688847 0.76 TAAR1 (0.41) HTR2AHTR1AHTR6
SCHEMBL31618142 0.74 CYP2C9 (0.54) AOC3HTR2AHTR1AHTR6
SCHEMBL1710455 0.73 ALDH1A1 (0.50) ACHE
SCHEMBL1014275 0.73 ALDH1A1 (0.50) ACHE
SCHEMBL2937482 0.72 AOC3 (0.73) AOC3HTR2AHTR1AHTR6
SCHEMBL9689684 0.71 NOS1 (0.43) AOC3HTR2AHTR1ANOS1HTR6
SCHEMBL9689679 0.71 HTR6 (0.45) AOC3HTR2AHTR1ANOS1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed