SCHEMBL9701397

SCHEMBL9701397

COc1ccc(CC2CNc3c(N)cc(Br)cc3CN2CC=C(C)C)cc1OC

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.33
CA2 P00918 4/20 0.33
CA9 Q16790 4/20 0.33
CA12 O43570 2/20 0.33
LMNA P02545 3/20 0.33
ALDH1A1 P00352 4/20 0.33
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP2D6 P10635 1/20 0.32
HTT P42858 2/20 0.32
GLA P06280 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702570 0.59 MAPT (0.42) LMNAALDH1A1KDM4EMAPK1HTT
SCHEMBL11057207 0.59 DRD2 (0.69) LMNAALDH1A1KDM4EMAPK1HSD17B10
SCHEMBL11157667 0.57 ALDH1A1 (0.55) CA1CA2CA9CA12LMNA
SCHEMBL14412911 0.57 MAPK1 (0.46) CA1CA2CA9CA12LMNA
SCHEMBL7902351 0.56 OPRM1 (0.34) KDM4E
SCHEMBL3367454 0.55 CA2 (0.59) CA1CA2CA9CA12LMNA
SCHEMBL11373073 0.55 CHRNB4 (0.56) CA1CA2CA9CA12LMNA
SCHEMBL14421411 0.55 CHRNB4 (0.56) CA1CA2CA9CA12LMNA
SCHEMBL7902097 0.55 SIGMAR1 (0.34)
SCHEMBL29910924 0.54 CA2 (0.58) CA1CA2CA9CA12MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992013860-A1 NEW 4,5,6,7-TETRAHYDRO-IMIDAZO-[4,5,lJK][1,4]-BENZODIAZEPINE-2-(1H)-THIONES, A METHOD OF PREPARING THEM AS WELL AS DRUGS CONTAINING THEM, AND INTERMEDIATES FOR THE PREPARATION OF THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-08-20 WO disclosed