SCHEMBL9704539

SCHEMBL9704539

COc1cc([S+](C)[O-])ccc1-c1nc2cc3c(=O)[nH]c(C)c(C)c3cc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 9/20 0.40
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
PDE5A O76074 1/20 0.36
CDK4 P11802 1/20 0.35
CCNA2 P20248 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35
CCND3 P30281 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
ERAP1 Q9NZ08 1/20 0.34
GUSB P08236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703323 0.84 CDK4 (0.47) AMY1APDE3BPDE3APDE5ACDK4
SCHEMBL9703649 0.82 AMY1A (0.43) AMY1APDE3BPDE3APDE5ATP53
SCHEMBL9703617 0.82 AMY1A (0.42) AMY1APDE3BPDE3APDE5ATP53
SCHEMBL9704436 0.80 PDE5A (0.43) AMY1APDE3BPDE3APDE5ANPC1
SCHEMBL9704521 0.80 CDK4 (0.42) AMY1APDE3BPDE3APDE5ACDK4
SCHEMBL9705442 0.79 KDM4E (0.41) AMY1APDE3BPDE3APDE5A
SCHEMBL9702924 0.78 AMY1A (0.41) AMY1APDE3BPDE3APDE5ATP53
SCHEMBL10852513 0.77 AMY1A (0.40) AMY1APDE3BPDE3APDE5ATP53
SCHEMBL10551908 0.77 AMY1A (0.39) AMY1APDE3BPDE3APDE5ATP53
SCHEMBL10700314 0.76 AMY1A (0.48) AMY1APDE3BPDE3ATP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed
EP-0275888-A2 Tricyclic benzimidazoles, process for their preparation and use as medicaments Roche Diagnostics GmbH (DE) 1988-07-27 EP disclosed