SCHEMBL9707736

SCHEMBL9707736

CC(C)Cn1c(=O)[nH]c2nc(C(C)C)n(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.42
ADORA2B P29275 2/20 0.42
USP1 O94782 8/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
ADORA1 P30542 1/20 0.35
PPARG P37231 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708314 0.92 ADORA2B (0.38) ADORA3ADORA2BUSP1ADORA1PPARG
SCHEMBL9708424 0.91 ADORA2B (0.40) ADORA3ADORA2BUSP1ADORA1PPARG
SCHEMBL9708252 0.91 ADORA3 (0.42) ADORA3ADORA2BUSP1GRIN1GRIN2B
SCHEMBL9708226 0.90 AGTR1 (0.38) ADORA3ADORA2BUSP1PPARG
SCHEMBL9707407 0.90 GPR18 (0.39) USP1PPARG
SCHEMBL9707641 0.89 AGTR1 (0.42) ADORA3ADORA2B
SCHEMBL9708640 0.89 USP1 (0.42) USP1PPARG
SCHEMBL9707357 0.89 ADORA2A (0.41) ADORA3ADORA2BUSP1ADORA1PPARG
SCHEMBL9707560 0.88 PPARG (0.42) USP1PPARG
SCHEMBL9707522 0.88 AGTR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed