SCHEMBL9708314

SCHEMBL9708314

CCn1c(=O)[nH]c2nc(C(C)C)n(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.38
ADORA3 P0DMS8 2/20 0.38
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
USP1 O94782 4/20 0.38
PPARG P37231 4/20 0.37
AGTR1 P30556 2/20 0.37
AGTR2 P50052 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708424 0.93 ADORA2B (0.40) ADORA2BADORA3ADORA2AADORA1USP1
SCHEMBL9707736 0.92 ADORA3 (0.42) ADORA2BADORA3ADORA1USP1PPARG
SCHEMBL9708226 0.91 AGTR1 (0.38) ADORA2BADORA3USP1PPARGAGTR1
SCHEMBL9707407 0.90 GPR18 (0.39) USP1PPARGAGTR1AGTR2
SCHEMBL9707357 0.89 ADORA2A (0.41) ADORA2BADORA3ADORA2AADORA1USP1
SCHEMBL9708640 0.89 USP1 (0.42) USP1PPARG
SCHEMBL9707560 0.89 PPARG (0.42) USP1PPARGAGTR1AGTR2
SCHEMBL9708298 0.89 ADORA2B (0.40) ADORA2BADORA3ADORA2AADORA1AGTR1
SCHEMBL9707370 0.88 PPARG (0.36) USP1PPARGAGTR1AGTR2
SCHEMBL9707904 0.88 AGTR1 (0.45) ADORA2BADORA3ADORA2AADORA1AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed