SCHEMBL9709743

SCHEMBL9709743

CCc1cc(NCc2ccc(-c3ccccc3C3(C(c4ccccc4)(c4ccccc4)c4ccccc4)N=NN=N3)cc2)c2cc(C(=O)O)ccc2n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.41
AGTR2 P50052 8/20 0.41
IP6K1 Q92551 1/20 0.34
IP6K3 Q96PC2 1/20 0.34
IP6K2 Q9UHH9 1/20 0.34
VCP P55072 1/20 0.34
PTGFR P43088 1/20 0.33
SCD O00767 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709875 0.88 AGTR1 (0.42) AGTR1AGTR2
SCHEMBL9709729 0.79 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL9709687 0.73 CD38 (0.44) AGTR1AGTR2
SCHEMBL9709723 0.73 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL9709740 0.72 LTB4R2 (0.51) AGTR1AGTR2
SCHEMBL9660639 0.71 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9709700 0.70 VCP (0.52) AGTR1AGTR2VCPSCD
SCHEMBL9208929 0.69 PDK2 (0.42)
SCHEMBL9709698 0.68 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9489948 0.67 ATM (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed