SCHEMBL9727395

SCHEMBL9727395

O=C1CCCN1S(=O)(=O)c1ccccc1C1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 3/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 1/20 0.38
STAT3 P40763 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 1/20 0.37
DRD2 P14416 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
PTGS2 P35354 1/20 0.36
MGLL Q99685 1/20 0.36
ACLY P53396 1/20 0.36
HTR6 P50406 2/20 0.36
CNR1 P21554 1/20 0.36
ALDH1A1 P00352 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727446 0.99 MEN1 (0.41) KMT2AMEN1GAATSHRCYP3A4
SCHEMBL9727311 0.84 HTR6 (0.41) KMT2AMEN1GAATSHRLMNA
SCHEMBL9727392 0.74 LMNA (0.59) KMT2AMEN1GAATSHRLMNA
SCHEMBL9727442 0.72 LMNA (0.61) KMT2AMEN1GAATSHRLMNA
SCHEMBL10179999 0.72 HSD11B1 (0.48) KMT2AMEN1GAAPTGS2HTR6
SCHEMBL7380549 0.72 PKM (0.62) KMT2AMEN1GAACYP3A4CYP2C9
SCHEMBL10180538 0.71 PTGS2 (0.49) GAATSHRCYP3A4CYP2C9CYP2C19
SCHEMBL10877910 0.71 CHRM4 (0.53) KMT2AMEN1TSHRCYP3A4CYP2C9
SCHEMBL10876708 0.71 CYP2C9 (0.49) KMT2AMEN1GAATSHRCYP3A4
SCHEMBL10879279 0.71 GAA (0.50) KMT2AMEN1GAATSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed
EP-0335758-A2 Derivatives of 1-arylsulfonyl-2-pyrolidinone, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1989-10-04 EP disclosed