SCHEMBL9727667

SCHEMBL9727667

COc1ccc(CC2Oc3cc(CCCO)c(O[Si](C)(C)C(C)(C)C)cc3C2C)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
ALOX5 P09917 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
DRD2 P14416 1/20 0.32
TNKS2 Q9H2K2 1/20 0.31
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9843450 0.86 DRD2 (0.31) NPSR1DRD2
SCHEMBL9727737 0.71 ESR1 (0.42)
SCHEMBL9727495 0.68 ALDH1A1 (0.43) CYP3A4EDNRBEDNRA
SCHEMBL9727708 0.68 ALDH1A1 (0.42) CYP3A4ALOX5
SCHEMBL4654931 0.66 DRD2 (0.46) DRD2
SCHEMBL9727705 0.65 ABCB1 (0.41) CYP3A4DRD2
SCHEMBL9727728 0.65 NR1I2 (0.32)
SCHEMBL2675281 0.65 PPARA (0.53) CYP3A4CYP11B1CYP11B2
SCHEMBL8503579 0.64 SLC6A2 (0.38) DRD2TNKS2
SCHEMBL7631655 0.63 DRD2 (0.48) CYP3A4POLBDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed