SCHEMBL9733462

SCHEMBL9733462

Cn1c(Cc2ccccc2F)nnc1C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
ESR2 Q92731 1/20 0.48
ACHE P22303 1/20 0.42
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 2/20 0.42
TSHR P16473 2/20 0.40
MAOB P27338 1/20 0.40
PARP15 Q460N3 1/20 0.40
PARP14 Q460N5 1/20 0.40
PARP10 Q53GL7 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PLK1 P53350 1/20 0.37
PDE3B Q13370 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735004 0.86 CA5A (0.44) GAAESR2ALDH1A1KDM4E
SCHEMBL9733754 0.81 ALDH1A1 (0.44) GAAESR2ALDH1A1KDM4ETSHR
SCHEMBL25586552 0.81 PKM (0.49) ALDH1A1HPGDLMNAPKMMEN1
SCHEMBL16798247 0.74 ALDH1A1 (0.42) GAAESR2ALDH1A1KDM4EMAOB
SCHEMBL9734773 0.70 GAA (0.41) GAAALDH1A1KDM4ELMNAPKM
SCHEMBL9733514 0.69 CA5A (0.42) GAAESR2ALDH1A1KDM4ETSHR
SCHEMBL3461564 0.68 MAPK8 (0.49) GAAALDH1A1KDM4ETSHRMAOB
SCHEMBL30091602 0.68 ALDH1A1 (0.42) ALDH1A1KDM4EMAOBPARP15PARP14
SCHEMBL9734745 0.68 BRD4 (0.39) KDM4ENPSR1LMNAPKMHSD17B10
SCHEMBL3571510 0.68 GUCY1A1 (0.54) GAAESR2ALDH1A1KDM4EMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US claimed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US claimed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP claimed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP claimed
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed