SCHEMBL9735004

SCHEMBL9735004

Cn1c(Cc2c(F)cccc2F)nnc1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.44
GAA P10253 1/20 0.36
ESR2 Q92731 1/20 0.36
TP53 P04637 1/20 0.35
CD38 P28907 1/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPK8 P45983 1/20 0.34
JAK2 O60674 3/20 0.34
JAK1 P23458 3/20 0.34
JAK3 P52333 3/20 0.34
ROCK2 O75116 2/20 0.34
GRK2 P25098 2/20 0.34
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
ADORA1 P30542 1/20 0.34
GLS O94925 1/20 0.33
TYK2 P29597 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733462 0.86 GAA (0.48) GAAESR2ALDH1A1KDM4E
SCHEMBL9734773 0.84 GAA (0.41) CA5AGAATP53ALDH1A1ROCK2
SCHEMBL9733514 0.83 CA5A (0.42) CA5AGAAESR2TP53CD38
SCHEMBL9734745 0.81 BRD4 (0.39) TP53ROCK2GRK2ADORA2AADORA2B
SCHEMBL9733899 0.81 ALDH1A1 (0.42) GAAALDH1A1KDM4E
SCHEMBL9733613 0.81 GRK2 (0.36) CA5AGAAESR2TP53ALDH1A1
SCHEMBL9734947 0.77 ALDH1A1 (0.38) CA5ATP53ALDH1A1ROCK2GRK2
SCHEMBL9733488 0.70 DHODH (0.37) CA5ATP53ALDH1A1
SCHEMBL9734269 0.69 ALDH1A1 (0.41) GAATP53ALDH1A1ADORA2AADORA2B
SCHEMBL9733754 0.68 ALDH1A1 (0.44) GAAESR2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US claimed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US claimed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP claimed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP claimed
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed