SCHEMBL9734773

SCHEMBL9734773

CNC(=O)c1nnc(Cc2c(F)cccc2F)n1C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
TP53 P04637 1/20 0.39
GRK2 P25098 3/20 0.37
ROCK2 O75116 2/20 0.37
HDAC6 Q9UBN7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ACSS2 Q9NR19 1/20 0.35
CA5A P35218 1/20 0.35
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.34
PKM P14618 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 2/20 0.33
EGFR P00533 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733613 0.88 GRK2 (0.36) GAATP53GRK2ROCK2HDAC6
SCHEMBL9734745 0.88 BRD4 (0.39) TP53GRK2ROCK2HDAC6L3MBTL1
SCHEMBL9735004 0.84 CA5A (0.44) GAATP53GRK2ROCK2CA5A
SCHEMBL9733899 0.80 ALDH1A1 (0.42) GAAL3MBTL1LMNAKMT2AALDH1A1
SCHEMBL25586082 0.78 HDAC6 (0.52) GAAHDAC6LMNAPKMMAPK1
SCHEMBL9734947 0.76 ALDH1A1 (0.38) TP53GRK2ROCK2CA5AALDH1A1
SCHEMBL9733514 0.71 CA5A (0.42) GAATP53CA5AKMT2AALDH1A1
SCHEMBL9733462 0.70 GAA (0.48) GAALMNAPKMKMT2AALDH1A1
SCHEMBL25586090 0.69 HDAC6 (0.51) HDAC6LMNAPKMMAPK1KMT2A
SCHEMBL9734269 0.69 ALDH1A1 (0.41) GAATP53L3MBTL1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US claimed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US claimed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP claimed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP claimed
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed