SCHEMBL9734745

SCHEMBL9734745

CCNC(=O)c1nnc(Cc2c(F)cccc2F)n1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.39
GRK2 P25098 4/20 0.38
ROCK2 O75116 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
ATM Q13315 1/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
PRKCA P17252 1/20 0.35
GRK5 P34947 1/20 0.35
GRK1 Q15835 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TP53 P04637 1/20 0.34
PDE2A O00408 1/20 0.34
PDE10A Q9Y233 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734773 0.88 GAA (0.41) GRK2ROCK2L3MBTL1ADORA2AADORA2B
SCHEMBL9733613 0.85 GRK2 (0.36) GRK2ROCK2L3MBTL1ATMLMNA
SCHEMBL9735004 0.81 CA5A (0.44) GRK2ROCK2ADORA2AADORA2BADORA1
SCHEMBL9733899 0.80 ALDH1A1 (0.42) L3MBTL1LMNAKDM4ENPSR1HSD17B10
SCHEMBL9734947 0.73 ALDH1A1 (0.38) GRK2ROCK2ADORA2AADORA2BADORA1
SCHEMBL9733514 0.71 CA5A (0.42) ADORA2AADORA2BADORA1KDM4ETP53
SCHEMBL13226271 0.70 RAB9A (0.57) ATM
SCHEMBL9734269 0.68 ALDH1A1 (0.41) L3MBTL1ADORA2AADORA2BADORA1KDM4E
SCHEMBL9733462 0.68 GAA (0.48) LMNAPKMKDM4ENPSR1HSD17B10
SCHEMBL9733754 0.67 ALDH1A1 (0.44) L3MBTL1LMNAMAPK1KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP claimed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP claimed
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed