SCHEMBL9733727

SCHEMBL9733727

CC1(C)C=C(n2ccccc2=S)c2cc(Br)ccc2C1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
PGR P06401 1/20 0.31
CHRM1 P11229 1/20 0.31
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
APOBEC3G Q9HC16 1/20 0.30
ALDH1A1 P00352 1/20 0.30
PPARG P37231 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
NCOR2 Q9Y618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733913 0.85 TDP1 (0.37) PDE4BL3MBTL1TDP1
SCHEMBL9733966 0.82 ALDH1A1 (0.33) PGRTSHRALDH1A1
SCHEMBL9733353 0.81 CHRM1 (0.37) L3MBTL1PGRCHRM1HPGDALDH1A1
SCHEMBL10433117 0.73 ESR1 (0.34) PDE4BL3MBTL1TDP1KDM4ETSHR
SCHEMBL9733434 0.70 SLC6A2 (0.39)
SCHEMBL9733018 0.70 HRH4 (0.34) L3MBTL1PGRALDH1A1PPARGNPSR1
SCHEMBL9733195 0.68 HRH4 (0.34)
SCHEMBL9733614 0.68 ALDH1A1 (0.35) ALDH1A1RXFP1
SCHEMBL9734559 0.68 RXFP1 (0.39) L3MBTL1KDM4ETSHRALDH1A1PPARG
SCHEMBL9733797 0.68 MEN1 (0.40) TDP1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed