SCHEMBL9734404

SCHEMBL9734404

CC(=O)Nc1ccc2c(c1)C(n1ccccc1=O)=CC(C)(C)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.43
CYP1A2 P05177 1/20 0.43
ADRA2A P08913 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2C P28335 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR2B P41595 1/20 0.43
ALDH1A1 P00352 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
F10 P00742 1/20 0.41
PDK2 Q15119 2/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSP90AA1 P07900 1/20 0.38
TLR9 Q9NR96 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733318 0.85 S100A4 (0.38) NPC1RAB9AMAPTF10PDK2
SCHEMBL9733434 0.82 SLC6A2 (0.39) SLC6A2SLC6A4MEN1KMT2AF10
SCHEMBL9734695 0.81 KMT2A (0.40) ALDH1A1MEN1KMT2AMAPTF10
SCHEMBL10433122 0.80 F10 (0.40) ALDH1A1SMN1; SMN2F10PDK2KDM4E
SCHEMBL10433092 0.80 F10 (0.36) F10
SCHEMBL9733913 0.79 TDP1 (0.37) SLC6A2SLC6A4MEN1KMT2ARAB9A
SCHEMBL9733018 0.79 HRH4 (0.34) SLC6A2SLC6A4ALDH1A1L3MBTL1
SCHEMBL9734559 0.78 RXFP1 (0.39) HTR2CHTR2BALDH1A1MEN1KMT2A
SCHEMBL8085176 0.78 MAOA (0.42) MAOACYP1A2ADRA2ASLC6A2HTR2C
SCHEMBL9733614 0.77 ALDH1A1 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed