SCHEMBL9734947

SCHEMBL9734947

Cn1c(CO)nnc1Cc1c(F)cccc1F

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
AR P10275 1/20 0.35
ADORA2A P29274 3/20 0.34
ADORA2B P29275 3/20 0.34
ADORA1 P30542 1/20 0.34
MAPT P10636 1/20 0.34
CA5A P35218 1/20 0.33
NOTUM Q6P988 1/20 0.33
PCSK9 Q8NBP7 1/20 0.33
POLB P06746 1/20 0.33
TP53 P04637 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
ROCK2 O75116 1/20 0.32
GRK2 P25098 1/20 0.32
HPGD P15428 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735004 0.77 CA5A (0.44) ALDH1A1ADORA2AADORA2BADORA1CA5A
SCHEMBL9734773 0.76 GAA (0.41) ALDH1A1ADORA2AADORA2BCA5APOLB
SCHEMBL9733899 0.73 ALDH1A1 (0.42) ALDH1A1MAPTPOLBHPGDNPC1
SCHEMBL9733613 0.73 GRK2 (0.36) ALDH1A1CA5ATP53ROCK2GRK2
SCHEMBL9734745 0.73 BRD4 (0.39) ADORA2AADORA2BADORA1TP53ROCK2
SCHEMBL22894792 0.67 PPARG (0.40) MAPTPOLBTP53NPC1RAB9A
SCHEMBL113326 0.66 TAAR1 (0.48) ALDH1A1MAPTPOLBTAAR1NPC1
SCHEMBL9733514 0.66 CA5A (0.42) ALDH1A1ADORA2AADORA2BADORA1MAPT
SCHEMBL5205493 0.66 TAAR1 (0.46) ALDH1A1ARPOLBTP53TAAR1
SCHEMBL3648972 0.63 HDAC6 (0.52) TP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed