SCHEMBL9733899

SCHEMBL9733899

CCOC(=O)c1nnc(Cc2c(F)cccc2F)n1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
KDM4E B2RXH2 4/20 0.42
RAB9A P51151 2/20 0.41
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41
MAPT P10636 3/20 0.40
HTT P42858 1/20 0.40
CYP1A2 P05177 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
ALOX15 P16050 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 3/20 0.38
TSHR P16473 3/20 0.38
GLA P06280 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733754 0.87 ALDH1A1 (0.44) ALDH1A1KDM4ERAB9AMAPTSMN1; SMN2
SCHEMBL9734269 0.86 ALDH1A1 (0.41) ALDH1A1KDM4EPTGESALOX5MAPT
SCHEMBL9735004 0.81 CA5A (0.44) ALDH1A1KDM4EGAA
SCHEMBL9734773 0.80 GAA (0.41) ALDH1A1KDM4EKMT2AGAAPOLB
SCHEMBL9734745 0.80 BRD4 (0.39) KDM4EHSD17B10NPSR1L3MBTL1LMNA
SCHEMBL9733669 0.77 ALDH1A1 (0.48) ALDH1A1KDM4ERAB9APTGESALOX5
SCHEMBL9733613 0.77 GRK2 (0.36) ALDH1A1RAB9AKMT2ANPC1MEN1
SCHEMBL9734321 0.76 MAPT (0.46) ALDH1A1KDM4EMAPTTDP1SMN1; SMN2
SCHEMBL9734947 0.73 ALDH1A1 (0.38) ALDH1A1RAB9AMAPTSMN1; SMN2NPC1
SCHEMBL17324355 0.72 PTGES (0.48) ALDH1A1KDM4ERAB9APTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed