SCHEMBL9737862

SCHEMBL9737862

CCCN(CCC)C(=O)Cc1c(-c2ccc(Cl)cc2)nn2cccnc12

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSPO P30536 4/20 0.52
GMNN O75496 1/20 0.50
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50
CYP3A4 P08684 1/20 0.50
BLM P54132 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
NR1I2 O75469 1/20 0.49
ABCB11 O95342 1/20 0.49
ALB P02768 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADORA1 P30542 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
OPRK1 P41145 1/20 0.49
PDE4D Q08499 1/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738542 0.93 TSPO (0.44) TSPOGMNNLMNAPOLBCYP3A4
SCHEMBL9737796 0.91 GABRA2 (0.47)
SCHEMBL9737961 0.87 ALDH1A1 (0.43) TSPO
SCHEMBL9737606 0.84 KDM4E (0.49) LMNA
SCHEMBL9737634 0.83 KDM4E (0.48)
SCHEMBL18116342 0.82 HTR1B (0.44) TSPOLMNA
SCHEMBL9738192 0.82 KDM4E (0.39)
SCHEMBL9738434 0.81 KCNQ3 (0.41) LMNA
SCHEMBL9737572 0.80 TSPO (0.45) TSPOLMNACYP3A4ALBOPRK1
SCHEMBL9738747 0.78 ALDH1A1 (0.45) TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114944-A Anxiolytic and anticonvulsant agents; muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1992-05-19 US claimed