SCHEMBL9738542

SCHEMBL9738542

CCCN(CCC)C(=O)Cc1c(-c2ccc(C)cc2)nn2cccnc12

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSPO P30536 2/20 0.44
HTR1B P28222 1/20 0.42
HTR2B P41595 1/20 0.42
GMNN O75496 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
BLM P54132 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737862 0.93 TSPO (0.52) TSPOGMNNLMNAPOLBCYP3A4
SCHEMBL9737796 0.92 GABRA2 (0.47)
SCHEMBL9737572 0.88 TSPO (0.45) TSPOHTR1BHTR2BLMNACYP3A4
SCHEMBL9737163 0.84 ALDH1A1 (0.43) LMNANPSR1
SCHEMBL9737283 0.84 PTGDR2 (0.47) LMNAPOLB
SCHEMBL18116342 0.83 HTR1B (0.44) TSPOHTR1BHTR2BLMNA
SCHEMBL9737491 0.83 PTGS2 (0.41) NPSR1
SCHEMBL9737185 0.81 KCNQ3 (0.41)
SCHEMBL9737961 0.79 ALDH1A1 (0.43) TSPO
SCHEMBL9738747 0.78 ALDH1A1 (0.45) TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114944-A Anxiolytic and anticonvulsant agents; muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1992-05-19 US claimed
US-5114944-A Anxiolytic and anticonvulsant agents; muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1992-05-19 US disclosed