SCHEMBL9742145

SCHEMBL9742145

CCCc1cc(Cl)c(SC(=O)N(C)C)c(C(C)=O)c1OC(C)=O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.35
ALOX5 P09917 2/20 0.34
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30
ABCB11 O95342 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10553104 0.78 PRKCI (0.35) PRKCIALOX5ALDH1A1KDM4EHPGD
SCHEMBL9747175 0.69 PRKCI (0.42) PRKCIALOX5ALDH1A1KDM4EHPGD
SCHEMBL9027495 0.68 PTPN1 (0.50) PRKCIALOX5KDM4EHSD17B10PPARG
SCHEMBL9029445 0.66 ALOX5 (0.60) PRKCIALOX5ALDH1A1KDM4ESMN1; SMN2
SCHEMBL13116411 0.65 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9739521 0.65 PRKCI (0.56) PRKCIALOX5ALDH1A1KDM4EHPGD
SCHEMBL17804010 0.63 ALDH1A1 (0.36) ALDH1A1KDM4EHPGD
SCHEMBL13116342 0.63 CA2 (0.35) ALDH1A1KDM4EHPGD
SCHEMBL9740854 0.62 PRKCI (0.51) PRKCIALOX5KDM4EHPGD
SCHEMBL2924582 0.62 THRB (0.39) ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087638-A Inhibitors of mammalian leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1992-02-11 US disclosed
EP-0338782-A1 Benzofuran derivatives MERCK FROSST CANADA INC. (CA) 1989-10-25 EP disclosed
US-4863958-A TREATING ALLERGIC CONDITIONS, ASTHMA, CARDIOVASCULAR DISORDERS, AND INFLAMMATION MERCK FROSST CANADA, INC. (CA) 1989-09-05 US disclosed