SCHEMBL9749287

SCHEMBL9749287

Cc1c(Oc2ccc(F)cc2)ccnc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 2/20 0.41
KDR P35968 2/20 0.41
TRPA1 O75762 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
KCNH2 Q12809 2/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
MET P08581 4/20 0.39
MRGPRX1 Q96LB2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AXL P30530 3/20 0.37
RET P07949 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293301 0.76 HSPB1 (0.43) KCNH2MRGPRX1HTR2AL3MBTL1ALDH1A1
SCHEMBL6149796 0.74 ALDH1A1 (0.44) TRPA1CYP3A4L3MBTL1ALDH1A1LMNA
SCHEMBL17508484 0.73 TRPA1 (0.42) PDGFRAKDRTRPA1CYP1A2CYP3A4
SCHEMBL17524535 0.71 TRPA1 (0.40) PDGFRAKDRTRPA1CYP1A2CYP3A4
SCHEMBL3586415 0.71 TRPA1 (0.37) PDGFRAKDRTRPA1CYP1A2CYP3A4
SCHEMBL9343291 0.70 TGFBR1 (0.44) TRPA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7470310 0.70 MAOA (0.38) PDGFRAKDRTRPA1CYP1A2CYP3A4
SCHEMBL17524357 0.69 TRPA1 (0.50) TRPA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14285766 0.68 RET (0.44) PDGFRAKDRTRPA1CYP1A2CYP3A4
SCHEMBL7463159 0.68 RET (0.44) PDGFRAKDRTRPA1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114955-A Derivatives with pyridine as gastrointestinal disorders and antisecretory agents HOECHST AKETIENGESELLSCHAFT (DE) 1992-05-19 US disclosed