SCHEMBL9753207

SCHEMBL9753207

Cc1cc(C)n2nc(C(C)C)c(C=O)c(-c3ccc(F)cc3)c12

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
GCGR P47871 10/20 0.39
PTGS2 P35354 3/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HMGCR P04035 1/20 0.35
MAPK10 P53779 1/20 0.34
MAPK14 Q16539 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753703 0.90 GCGR (0.36) ALDH1A1GCGRPTGS2NPC1RAB9A
SCHEMBL9753707 0.90 GCGR (0.36) ALDH1A1GCGRPTGS2NPC1RAB9A
SCHEMBL9753393 0.86 HMGCR (0.38) ALDH1A1GCGRPTGS2HMGCR
SCHEMBL9752903 0.82 MAPK14 (0.43) ALDH1A1GCGRPTGS2NPC1RAB9A
SCHEMBL27346853 0.82 PPARA (0.41) ALDH1A1GCGRPTGS2NPC1RAB9A
SCHEMBL9753342 0.81 GCGR (0.55) GCGR
SCHEMBL9752971 0.81 PTGS2 (0.39) ALDH1A1PTGS2NPC1RAB9ASMN1; SMN2
SCHEMBL9753077 0.78 ALDH1A1 (0.44) ALDH1A1GCGRNPC1RAB9ASMN1; SMN2
SCHEMBL9753784 0.78 HMGCR (0.47) ALDH1A1HMGCR
SCHEMBL9753373 0.78 HMGCR (0.60) ALDH1A1PTGS2HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed
CN-1056690-A PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO (JP) 1991-12-04 CN disclosed