SCHEMBL9756685

SCHEMBL9756685

COc1ccc(C(=O)Oc2c(N3CCCC3)nc(N3CCCC3)nc2N2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
ALDH1A1 P00352 1/20 0.46
SLC2A1 P11166 1/20 0.45
GPR119 Q8TDV5 4/20 0.44
TLR9 Q9NR96 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
MAPK1 P28482 1/20 0.43
GALR2 O43603 1/20 0.42
GALR1 P47211 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GBA1 P04062 3/20 0.42
SLC6A7 Q99884 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9756677 0.90 KMT2A (0.47) SMN1; SMN2GPR119TLR9TLR7GBA1
SCHEMBL9756680 0.89 MEN1 (0.55) SMN1; SMN2MAPTGPR119TLR9TLR7
SCHEMBL9756638 0.89 GBA1 (0.49) GPR119TLR9TLR7GBA1ADORA2A
SCHEMBL9668922 0.81 GPR119 (0.43) MAPTLMNAALDH1A1GPR119TLR9
SCHEMBL9756679 0.80 GBA1 (0.55) TLR9TLR7GBA1
SCHEMBL9756696 0.77 GPR119 (0.45) MAPTLMNAALDH1A1GPR119TLR9
4-Methylbenzoic Acid SCHEMBL9671138 0.75 GBA1 (0.48) SMN1; SMN2GPR119TLR9TLR7GBA1
SCHEMBL5233751 0.73 L3MBTL1 (0.66) SMN1; SMN2MAPTLMNAALDH1A1GPR119
SCHEMBL1458624 0.73 L3MBTL1 (0.73) SMN1; SMN2MAPTLMNAALDH1A1GPR119
SCHEMBL28494646 0.73 MEN1 (0.67) SMN1; SMN2MAPTLMNAALDH1A1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991011453-A2 5-OXYGENATED-2,4,6-TRIAMINOPYRIMIDINES THE UPJOHN COMPANY (US) 1991-08-08 WO claimed