SCHEMBL9757518

SCHEMBL9757518

O=c1[nH]c2ccccc2n1C1CCN(CCCN2c3cccc4cccc(c34)S2(=O)=O)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.62
CYP2C9 P11712 1/20 0.62
CHRM1 P11229 5/20 0.60
DRD2 P14416 5/20 0.58
KCNH2 Q12809 4/20 0.58
PMP22 Q01453 2/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
ADRA1D P25100 2/20 0.56
ADRA1A P35348 2/20 0.56
ADRA1B P35368 1/20 0.56
HTR7 P34969 2/20 0.54
MEN1 O00255 1/20 0.53
SLC22A2 O15244 1/20 0.53
NR1I2 O75469 1/20 0.53
GMNN O75496 1/20 0.53
USP2 O75604 1/20 0.53
LMNA P02545 1/20 0.53
CYP1A2 P05177 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5984495 0.82 CYP2D6 (0.85) CYP2D6CYP2C9CHRM1DRD2KCNH2
SCHEMBL9872838 0.80 HTR7 (0.54) DRD2KCNH2ADRA1AADRA1BHTR7
SCHEMBL6404859 0.78 CHRM1 (0.88) CYP2D6CYP2C9CHRM1DRD2KCNH2
SCHEMBL5772590 0.78 CYP2D6 (1.00) CYP2D6CYP2C9CHRM1DRD2KCNH2
SCHEMBL9757165 0.77 HTR7 (0.66) DRD2KCNH2ADRA1AADRA1BHTR7
SCHEMBL6404540 0.77 PLD1 (0.81) CYP2D6CYP2C9CHRM1DRD2KCNH2
SCHEMBL11878362 0.77 ADRA1A (0.84) CYP2D6CYP2C9CHRM1DRD2KCNH2
SCHEMBL9757338 0.77 ADRA1D (0.60) ADRA1D
SCHEMBL11507088 0.77 DRD2 (0.82) CYP2D6CYP2C9CHRM1DRD2KCNH2
Hydrochloric Acid SCHEMBL7256214 0.77 CYP2D6 (0.76) CYP2D6CYP2C9CHRM1DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036075-A Serotonin antagonists RHONE-POULENC SANTE (FR) 1991-07-30 US disclosed
US-5021420-A Antiserotonine agents; central nervous system, gastroin-testinal and cardiovascular disorders RHONE-POULENC SANTE (FR) 1991-06-04 US disclosed