SCHEMBL9759024

SCHEMBL9759024

O=C([O-])COCCNc1cc(Oc2ccc(Cl)cc2Cl)ccc1[N+](=O)[O-].[Na+]

nearest known ligand 0.54

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.54
MAPT P10636 5/20 0.50
LMNA P02545 3/20 0.50
ALPG P10696 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTR6 P50406 1/20 0.42
PKM P14618 2/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
TTR P02766 1/20 0.41
PPOX P50336 1/20 0.41
PDE7A Q13946 1/20 0.39
S1PR4 O95977 1/20 0.39
FFAR1 O14842 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 2/20 0.37
SIRT5 Q9NXA8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9759305 0.90 TDP1 (0.58) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL9759130 0.88 MEN1 (0.58) TDP1MAPTLMNASMN1; SMN2KMT2A
SCHEMBL9759758 0.87 TDP1 (0.50) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL9759894 0.87 TDP1 (0.49) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL9760115 0.83 MEN1 (0.56) TDP1MAPTLMNASMN1; SMN2KMT2A
SCHEMBL10996617 0.83 TDP1 (0.59) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL10996710 0.81 TDP1 (0.62) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL9759962 0.80 MEN1 (0.43) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL11000498 0.80 TDP1 (0.60) TDP1MAPTLMNAALPGSMN1; SMN2
SCHEMBL11017180 0.80 MEN1 (0.61) TDP1MAPTLMNASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028732-A Herbicidally active amino diphenyl ethers ROHM AND HAAS COMPANY (US) 1991-07-02 US disclosed
EP-0130041-B1 NOVEL HERBICIDAL SUBSTITUTED PYRIDYL PHENYL AND DIPHENYL ETHERS, HERBICIDAL COMPOSITIONS CONTAINING THEM, PROCESSES FOR THE PREPARATION THEREOF AND THE USE THEREOF FOR COMBATING WEEDS ROHM AND HAAS COMPANY (US) 1988-01-13 EP disclosed
EP-0130041-A1 Novel herbicidal substituted pyridyl phenyl and diphenyl ethers, herbicidal compositions containing them, processes for the preparation thereof and the use thereof for combating weeds ROHM AND HAAS COMPANY (US) 1985-01-02 EP disclosed