SCHEMBL9764142

SCHEMBL9764142

O=CC1=C(c2ccc(F)cc2)c2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.51
PTGS1 P23219 3/20 0.51
MAPK14 Q16539 1/20 0.39
BCHE P06276 1/20 0.38
CES1 P23141 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
MAOA P21397 1/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16139564 0.71 CES1 (0.44) CES1MAOANPC1POLBPKM
SCHEMBL23975284 0.71 PTGS2 (0.40) PTGS2PTGS1ESR1ESR2
SCHEMBL21703736 0.70 PTGS2 (0.35) PTGS2PTGS1BCHECES1ESR1
SCHEMBL6209822 0.68 MAOA (0.43) BCHECES1SLC6A4SLC6A3MAOA
SCHEMBL21294262 0.68 THRB (0.46) PTGS1ESR1ESR2NPC1PKM
SCHEMBL31185872 0.67 PRKCB (0.49) SMN1; SMN2CYP2D6ALDH1A1HSD17B10LMNA
SCHEMBL2222606 0.66 XDH (0.51) PTGS2PTGS1SLC6A4SLC6A3POLB
SCHEMBL1480938 0.66 KDM4E (0.52) PTGS2PTGS1SLC6A4SLC6A3MAOA
SCHEMBL27375940 0.66 PNMT (0.47) PTGS2PTGS1NPC1TP53POLB
SCHEMBL18032688 0.64 CES1 (0.67) BCHECES1MAOAPOLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032590-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1991-07-16 US disclosed
US-5001255-A Idene analogs of mevalonolactone and derivatives thereof SANDOZ PHARM. CORP. (US) 1991-03-19 US disclosed
EP-0216785-B1 INDENE ANALOGS OF MEVALONOLACTONE AND DERIVATIVES THEREOF SANDOZ AG (CH) 1991-01-30 EP disclosed
US-4968681-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
EP-0317845-A2 Substituted hydroxyl amines BAYER AG (DE) 1989-05-31 EP disclosed
EP-0216785-A1 INDENE ANALOGS OF MEVALONOLACTONE AND DERIVATIVES THEREOF. SANDOZ AG (CH) 1987-04-08 EP disclosed
WO-1986003488-A1 INDENE ANALOGS OF MEVALONOLACTONE AND DERIVATIVES THEREOF SANDOZ AG (CH) 1986-06-19 WO disclosed