SCHEMBL9764499

SCHEMBL9764499

CC(=O)NCc1cccc(C#CCOCCCCCCNCc2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
MAPK1 P28482 1/20 0.45
BCHE P06276 4/20 0.43
ACHE P22303 4/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
P4HB P07237 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAOA P21397 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
CHRM2 P08172 1/20 0.39
MAOB P27338 1/20 0.39
SCN8A Q9UQD0 1/20 0.39
MITF O75030 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764480 0.77 MMP2 (0.43) KDM4EMAPK1BCHEACHEALDH1A1
SCHEMBL9318691 0.76 SLC2A1 (0.48) KDM4EBCHEMEN1ALDH1A1KMT2A
SCHEMBL9764451 0.74 SMN1; SMN2 (0.45) KDM4EMAPK1BCHEACHEMEN1
SCHEMBL9763136 0.74 DRD4 (0.47) KDM4EMAPK1BCHEP4HBNPSR1
SCHEMBL9763494 0.73 DRD2 (0.47) BCHEACHEMAOACHRM2ADRB2
SCHEMBL9764455 0.72 MAOA (0.40) KDM4EMAPK1BCHEACHEP4HB
SCHEMBL9764397 0.71 ACACB (0.43) MAPK1ALDH1A1GAA
SCHEMBL10465009 0.70 EPHX2 (0.51) KDM4EMEN1ALDH1A1KMT2AHDAC3
SCHEMBL10417690 0.70 MAOA (0.48) KDM4EMAPK1BCHEACHEMAOA
SCHEMBL9763151 0.70 BCHE (0.49) KDM4EMAPK1BCHEACHEP4HB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed