SCHEMBL9764455

SCHEMBL9764455

CN(c1ccc(C#CCOCCCCCCNCc2ccccc2)cc1)S(C)(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.40
CHRM2 P08172 1/20 0.39
SIGMAR1 Q99720 4/20 0.37
KDM4E B2RXH2 3/20 0.36
MAPK1 P28482 1/20 0.36
SCN8A Q9UQD0 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
BCHE P06276 3/20 0.35
ACHE P22303 3/20 0.35
MITF O75030 1/20 0.35
GAA P10253 1/20 0.35
MAOB P27338 1/20 0.35
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9763494 0.84 DRD2 (0.47) MAOACHRM2SIGMAR1BCHEACHE
SCHEMBL9764480 0.81 MMP2 (0.43) MAOACHRM2SIGMAR1KDM4EMAPK1
SCHEMBL9764451 0.78 SMN1; SMN2 (0.45) MAOAKDM4EMAPK1BCHEACHE
SCHEMBL9763136 0.76 DRD4 (0.47) MAOACHRM2KDM4EMAPK1BCHE
SCHEMBL9763710 0.73 SIGMAR1 (0.43) MAOACHRM2SIGMAR1DRD2DRD4
SCHEMBL9318691 0.73 SLC2A1 (0.48) MAOACHRM2KDM4EBCHEMAOB
SCHEMBL9764499 0.72 KDM4E (0.45) MAOACHRM2KDM4EMAPK1SCN8A
SCHEMBL9763021 0.71 AR (0.51) MAOACHRM2SIGMAR1KDM4EBCHE
SCHEMBL9764397 0.71 ACACB (0.43) MAPK1GAA
SCHEMBL10417690 0.70 MAOA (0.48) MAOACHRM2SIGMAR1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed