SCHEMBL9768675

SCHEMBL9768675

O=c1[nH]cc(-c2ccc(Cl)cc2)n1CCCl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.48
HPGD P15428 6/20 0.48
MAPT P10636 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
RXFP1 Q9HBX9 2/20 0.47
KDM4E B2RXH2 4/20 0.37
GAA P10253 3/20 0.37
CYP2C9 P11712 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
NPC1 O15118 1/20 0.36
TYMP P19971 1/20 0.35
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768587 0.85 ALDH1A1 (0.48) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL4500559 0.83 ALDH1A1 (0.48) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL11258178 0.80 APEX1 (0.52) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL9768576 0.76 ALDH1A1 (0.46) ALDH1A1HPGDMAPTKDM4EGAA
SCHEMBL28829027 0.76 ALDH1A1 (0.42) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL28828985 0.74 AVPR2 (0.41) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL28828981 0.74 AVPR2 (0.41) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL28828879 0.73 TSHR (0.50) ALDH1A1HPGDMAPTNPSR1KDM4E
SCHEMBL11126289 0.70 ALDH1A1 (0.69) ALDH1A1HPGDMAPTNPSR1RXFP1
SCHEMBL4496826 0.69 DRD2 (0.38) ALDH1A1HPGDMAPTNPSR1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5059601-A IMIDAZOLONE DERIVATIVES WITH ACTIVITY ON CENTRAL NERVOUS SYSTEM AND ANTIHYPERTENSIVE ACTIVITY, PREPARATION METHODS THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ISTITUTO LUSOFARMACO D'ITALIA S.P.A. (IT) 1991-10-22 US disclosed
EP-0379990-A1 Imidazolone derivatives with activity on central nervous system and antihypertensive activity, preparation methods thereof, and pharmaceutical compositions containing them ISTITUTO LUSO FARMACO D'ITALIA S.p.A. (IT) 1990-08-01 EP disclosed