SCHEMBL9770688

SCHEMBL9770688

COC(=O)c1sc2nc3c(F)cccc3c(=O)n2c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
TRPV4 Q9HBA0 2/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 1/20 0.39
GPR139 Q6DWJ6 2/20 0.38
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
TP53 P04637 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
GAA P10253 2/20 0.36
RECQL P46063 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695797 0.71 KDM4E (0.52) TRPV4ALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL10696499 0.71 PDE7A (0.39) TRPV4LMNAALDH1A1HPGDRAB9A
SCHEMBL10696506 0.71 ALDH1A1 (0.62) MEN1KMT2AALDH1A1HPGDRAB9A
SCHEMBL10695759 0.69 CYP1A1 (0.43) ADORA2AALDH1A1HPGDSMN1; SMN2RXFP1
SCHEMBL10694328 0.68 ELANE (0.42) LMNAALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL9770629 0.68 TNKS (0.42) ADORA2AALDH1A1HPGDSMN1; SMN2
SCHEMBL23532121 0.66 MEN1 (0.50) MEN1KMT2ALMNAMAPK1ALDH1A1
SCHEMBL10695331 0.66 PDE7A (0.43) LMNAALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10696216 0.66 PARP1 (0.44) LMNAGPR139ALDH1A1HPGDRAB9A
SCHEMBL9770496 0.65 CYP1A2 (0.43) MEN1KMT2ATRPV4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030727-A Reacting an anthronilide derivative with a thiazole derivative or a fluorozuinazolone with a neucleophile BASF AKTIENGESELLSCHAFT (DE) 1991-07-09 US disclosed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP disclosed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP disclosed