SCHEMBL9779491

SCHEMBL9779491

Cc1nc(-c2ccccc2)cc(-c2cccc(C#N)c2)c1NC(=O)CCl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.46
GRM5 P41594 2/20 0.44
MAPT P10636 2/20 0.44
F11 P03951 1/20 0.44
CTSA P10619 1/20 0.43
ADORA1 P30542 4/20 0.42
ADORA2B P29275 3/20 0.42
ADORA3 P0DMS8 1/20 0.42
PIN1 Q13526 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
USP2 O75604 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
PRKDC P78527 1/20 0.41
ATR Q13535 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779218 0.92 ADORA2A (0.44) ADORA2AGRM5MAPTF11CTSA
SCHEMBL9779661 0.82 ALDH1A1 (0.51) MAPTALDH1A1LMNASMN1; SMN2USP2
SCHEMBL9779414 0.81 F11 (0.43) ADORA2AGRM5MAPTF11CTSA
SCHEMBL9779395 0.80 TSHR (0.47) MAPTALDH1A1LMNASMN1; SMN2USP2
Morpholine SCHEMBL9779664 0.78 ADORA2A (0.44) ADORA2AF11CTSAADORA1ADORA2B
SCHEMBL9779442 0.77 F11 (0.54) ADORA2AF11ADORA1PIN1ALDH1A1
SCHEMBL9779192 0.73 ADORA2A (0.53) ADORA2AF11ADORA1ADORA2BATR
SCHEMBL10430923 0.72 GABRA1 (0.50) ADORA2AMAPTF11ADORA1ADORA2B
SCHEMBL9779393 0.72 ADORA3 (0.51) MAPTF11ADORA3PIN1ALDH1A1
SCHEMBL9779299 0.69 F11 (0.55) GRM5F11PIN1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037824-A Cardiotonic, antiischemic agents FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1991-08-06 US disclosed
EP-0387070-A2 N-Containing heterocyclic compounds, processes for the preparation thereof and composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-09-12 EP disclosed