SCHEMBL98201

SCHEMBL98201

CC[N]c1ccc(O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.45
NOS2 P35228 3/20 0.45
NOS1 P29475 2/20 0.45
S100B P04271 1/20 0.44
ESR1 P03372 5/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
LMNA P02545 3/20 0.42
CYP3A4 P08684 3/20 0.42
MAPT P10636 3/20 0.42
ALOX15 P16050 3/20 0.42
CA12 O43570 3/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA9 Q16790 3/20 0.42
ESR2 Q92731 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HIF1A Q16665 2/20 0.42
HSD17B10 Q99714 2/20 0.42
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767212 0.74 PLAU (0.52) LMNAMAPTCA2ALDH1A1NPC1
SCHEMBL1735291 0.74 NOS3 (0.44) NOS3NOS2NOS1ESR1LMNA
SCHEMBL4607389 0.74 NOS1 (0.44) NOS1ESR1MAPTALOX15ESR2
SCHEMBL6385307 0.74 NOS3 (0.44) NOS3NOS1ESR1LMNACA1
SCHEMBL10672526 0.73 TRPA1 (0.46) ESR1KMT2AMEN1LMNACYP3A4
Hydroquinone SCHEMBL6071932 0.73 LMNA (0.67) ESR1KMT2AMEN1LMNACYP3A4
Hydroquinone SCHEMBL11180188 0.73 LMNA (0.67) ESR1KMT2AMEN1LMNACYP3A4
Hydroquinone SCHEMBL3095350 0.73 LMNA (0.67) ESR1KMT2AMEN1LMNACYP3A4
SCHEMBL53706 0.72
SCHEMBL2306420 0.72 ALDH1A1 (0.46) KMT2AMEN1LMNACYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118307501-A Dihydrophenanthropyrrole compound, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-07-09 CN claimed
CN-118059113-A Application of anemonin B4 derivative in preparation of medicine for preventing and treating psoriasis 苏州大学 2024-05-24 CN claimed
CN-117567543-A Anemonin B4 derivative and preparation method and application thereof 苏州大学 2024-02-20 CN claimed
EP-2426139-A1 CXCR4 antagonist and use thereof Biokine Therapeutics Ltd. (IL) 2012-03-07 EP claimed
US-8017585-B2 CXCR4 antagonist and use thereof BIOKINE THERAPEUTICS LTD. (IL) 2011-09-13 US claimed
US-20090181897-A1 CXCR4 ANTAGONIST AND USE THEREOF BIOKINE THERAPEUTICS LTD. (IL) 2009-07-16 US claimed
US-20060264378-A1 Cxcr4 antagonist and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-11-23 US claimed
EP-1412328-B1 DOLASTATIN 10 DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-10-04 EP claimed
EP-1541585-A1 CXCR4 ANTAGONIST AND USE THEREOF Fujii, Nobutaka (JP) 2005-06-15 EP claimed
US-6737409-B2 FOR CANCER THERAPY HOFFMANN-LA ROCHE INC. 2004-05-18 US claimed
EP-1412328-A1 DOLASTATIN 10 DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2004-04-28 EP claimed
US-20030055002-A1 Dolastatin 10 derivatives HOFFMANN-LA ROCHE INC. 2003-03-20 US claimed
WO-2003008378-A1 DOLASTATIN 10 DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2003-01-30 WO claimed
CN-118307501-A Dihydrophenanthropyrrole compound, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-07-09 CN disclosed
CN-118126032-A Fluorescent probe and preparation method and application thereof 广州谱赛生物医学科技有限公司 2024-06-04 CN disclosed
CN-118059113-A Application of anemonin B4 derivative in preparation of medicine for preventing and treating psoriasis 苏州大学 2024-05-24 CN disclosed
US-6127538-A HYDROXYALKYLATION OF A TRIAMINO TRIAZINE DERIVATIVE HAVING AT LEAST ONE REACTIVE NITROGEN BY REACTING WHILE HEATING WITH AN ALKANEDIOL OR ITS ADDUCT IN THE PRESENCE OF HYDROGEN AND A METAL CATALYST; BY-PRODUCT INHIBITION NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-10-03 US disclosed
WO-2000018759-A1 PHENYLALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-04-06 WO disclosed
EP-0882720-A1 METHODS FOR MODIFYING 1,3,5-TRIAZINE DERIVATIVES NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1998-12-09 EP disclosed
EP-0760369-A1 PROCESS FOR ALKYLATING TRIAZINE DERIVATIVE NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1997-03-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181897-A1 CXCR4 ANTAGONIST AND USE THEREOF CXCR4, ACKR3, CXCR1 NOS3 3130/4885NOS2 3301/4885NOS1 3289/4885
US-20030055002-A1 Dolastatin 10 derivatives DAD1, DDOST, NPC1 NOS3 2959/4885NOS2 3259/4885NOS1 2592/4885
US-20060264378-A1 Cxcr4 antagonist and use thereof CXCR4, ACKR3, CXCR1 NOS3 3130/4885NOS2 3301/4885NOS1 3289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.