SCHEMBL9825874

SCHEMBL9825874

c1cnc(N2CCN(CCCCOc3cccc4ncccc34)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.54
HTR1A P08908 4/20 0.54
DRD3 P35462 4/20 0.54
DRD2 P14416 3/20 0.54
DRD1 P21728 3/20 0.54
HTR1D P28221 1/20 0.53
HTR1B P28222 1/20 0.53
HRH3 Q9Y5N1 9/20 0.53
ABCB1 P08183 2/20 0.53
DRD5 P21918 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HTR7 P34969 2/20 0.49
HTR6 P50406 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9826692 0.81 DRD2 (0.55) HTR2AHTR1ADRD3DRD2DRD1
SCHEMBL9183697 0.81 P2RX7 (0.59) HTR1AHTR1DHTR1BABCB1TDP1
SCHEMBL23412437 0.78 NCF1 (0.58) HTR1AHTR1DHTR1BTDP1MEN1
SCHEMBL9188044 0.77 ABCB1 (0.51) HTR2AHTR1AHTR1DHTR1BHRH3
SCHEMBL9181173 0.77 P2RX7 (0.57) HTR1ADRD3HTR1DHTR1BHRH3
SCHEMBL23412188 0.77 NCF1 (0.51) HTR1AHTR1DHTR1BTDP1MEN1
SCHEMBL9825914 0.76 HRH3 (0.57) HTR2AHTR1ADRD3DRD2DRD1
SCHEMBL23412378 0.75 MAPT (0.52) HTR1AHTR1DHTR1BTDP1MEN1
SCHEMBL26492991 0.75 HTR1A (0.65) HTR2AHTR1ADRD3DRD2DRD1
SCHEMBL26108581 0.75 HTR1A (0.65) HTR2AHTR1ADRD3DRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP disclosed
US-4803203-A SCHIZOPHRENIA, NEUOLEPTIC AGENTS WARNER-LAMBERT COMPANY (US) 1989-02-07 US disclosed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US disclosed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP disclosed