SCHEMBL9828848

SCHEMBL9828848

C=C(COCCCCCCCCCCCCCCCC)COC(=O)CBr

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
FAAH O00519 2/20 0.47
TSHR P16473 2/20 0.44
NAAA Q02083 1/20 0.43
PAM P19021 2/20 0.40
TRPA1 O75762 1/20 0.40
ALDH1A1 P00352 1/20 0.40
DGKA P23743 1/20 0.40
RAD52 P43351 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
EPHX1 P07099 1/20 0.38
MEN1 O00255 1/20 0.37
THRB P10828 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPT P10636 1/20 0.37
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828285 0.88 PAM (0.49) CES2FAAHTSHRNAAAPAM
SCHEMBL9828212 0.87 DGKA (0.51) CES2FAAHTSHRNAAAPAM
SCHEMBL9828178 0.87 DGKA (0.51) CES2FAAHTSHRNAAAPAM
Bromide SCHEMBL10768699 0.84 CES2 (0.37) CES2FAAHTSHRPAMRAD52
SCHEMBL20898183 0.81 CES2 (0.59) CES2TSHRNAAAALDH1A1MEN1
SCHEMBL20898213 0.81 CES2 (0.59) CES2TSHRNAAAALDH1A1MEN1
SCHEMBL11415281 0.79 CES2 (0.56) CES2TSHRALDH1A1MEN1THRB
SCHEMBL9828659 0.79 ACHE (0.49) CES2FAAHEPHX1
SCHEMBL20896970 0.78 FAAH (0.59) CES2FAAHTSHRNAAATRPA1
SCHEMBL1032849 0.78 FAAH (0.59) CES2FAAHTSHRNAAATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0247201-B1 PROPANE-1,3-DIOL DERIVATIVES, A METHOD FOR THEIR PRODUCTION AND A PHARMACEUTICAL COMPOSITION LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1991-05-15 EP disclosed
US-4945098-A Novel propane-1,3-diol derivatives and use LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1990-07-31 US disclosed
EP-0247201-A1 PROPANE-1,3-DIOL DERIVATIVES, A METHOD FOR THEIR PRODUCTION AND A PHARMACEUTICAL COMPOSITION. LEO PHARM PROD LTD (DK) 1987-12-02 EP disclosed
WO-1987003281-A1 PROPANE-1,3-DIOL DERIVATIVES, A METHOD FOR THEIR PRODUCTION AND A PHARMACEUTICAL COMPOSITION LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 1987-06-04 WO disclosed