SCHEMBL9829358

SCHEMBL9829358

CCC(=O)Cn1ncc(-c2ccc(OC)cc2)nc1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
GRIN2B Q13224 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
ADORA2B P29275 1/20 0.42
MEN1 O00255 2/20 0.41
MAPT P10636 5/20 0.40
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KMT2A Q03164 3/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828154 0.87 LMNA (0.46) CHEK1ADORA3MEN1MAPTRAB9A
SCHEMBL9828844 0.85 CHEK1 (0.50) CHEK1MEN1MAPTRAB9ANPC1
SCHEMBL9829354 0.84 CHEK1 (0.43) CHEK1ADORA3MEN1MAPTRAB9A
SCHEMBL9829126 0.82 CHEK1 (0.40) CHEK1ADORA3ADORA2BMEN1MAPT
SCHEMBL9828939 0.82 MGAM (0.47) CHEK1MEN1MAPTRAB9ANPC1
SCHEMBL9828617 0.81 ALDH1A1 (0.51) CHEK1MEN1MAPTRAB9ANPC1
SCHEMBL9828641 0.78 MAPT (0.47) MEN1MAPTRAB9AALDH1A1HPGD
SCHEMBL9827533 0.78 NPC1 (0.46) GRIN2BADORA3MEN1MAPTRAB9A
SCHEMBL9832501 0.78 TLR8 (0.51) CHEK1MAPTRAB9ANPC1ALDH1A1
SCHEMBL9829232 0.74 FYN (0.44) CHEK1MEN1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233804-B1 MONOARYL-5-AS TRIAZINONES SUBSTITUTED IN POSITION 2, PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL PREPARATIONS PIERRE FABRE MEDICAMENT (FR) 1991-09-25 EP claimed