SCHEMBL9836237

SCHEMBL9836237

O=C(CCl)NC1c2ccccc2OCc2ncccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
P2RX7 Q99572 12/20 0.38
MAPT P10636 2/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836562 0.83 P2RX7 (0.36) ALDH1A1LMNAP2RX7MAPTCYP3A4
SCHEMBL9835913 0.82 P2RX7 (0.36) LMNASMN1; SMN2P2RX7MAPT
SCHEMBL9836786 0.81 DRD2 (0.43) ALDH1A1HTTSMN1; SMN2CYP2C19
SCHEMBL9836629 0.74 CYP2C19 (0.41) ALDH1A1LMNACYP1A2CYP2C19
SCHEMBL9836996 0.73 MAOA (0.48) LMNASMN1; SMN2P2RX7MAPTCYP1A2
SCHEMBL8797476 0.73 MAPT (0.43) ALDH1A1LMNASMN1; SMN2P2RX7MAPT
SCHEMBL9835161 0.72 HRH3 (0.38)
SCHEMBL9834971 0.72 ALDH1A1 (0.36) ALDH1A1
SCHEMBL9835174 0.72 MAPK14 (0.38) ALDH1A1SMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL9835877 0.71 GRIN1 (0.42) ALDH1A1LMNASMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP disclosed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US disclosed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP disclosed