SCHEMBL9836609

SCHEMBL9836609

c1ccc2c(c1)OCc1ncccc1C2NCCN1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HPGDS O60760 1/20 0.39
SLC40A1 Q9NP59 1/20 0.38
LMNA P02545 2/20 0.38
HIF1A Q16665 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CXCR4 P61073 1/20 0.38
MITF O75030 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
SMARCA2 P51531 1/20 0.38
MKNK1 Q9BUB5 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835161 0.91 HRH3 (0.38)
SCHEMBL9836629 0.77 CYP2C19 (0.41) MEN1KMT2AKDM4ELMNACYP1A2
SCHEMBL9834971 0.76 ALDH1A1 (0.36) MEN1KMT2A
SCHEMBL9835877 0.75 GRIN1 (0.42) LMNACYP3A4CYP2D6CXCR4
SCHEMBL9834568 0.75 HSP90AA1 (0.38) CYP3A4
SCHEMBL11112310 0.74 CYP3A4 (0.45) MEN1KMT2ACYP3A4POLB
SCHEMBL9835639 0.74 ALDH1A1 (0.42) CYP2D6POLB
SCHEMBL9836786 0.71 DRD2 (0.43) MEN1KMT2A
SCHEMBL9836237 0.70 ALDH1A1 (0.41) LMNACYP1A2CYP3A4
SCHEMBL9836619 0.70 CXCR4 (0.42) MEN1KMT2AL3MBTL1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US claimed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP claimed